Michael Humphreys, MD

PROF EMERITUS(WOS)

Dr. Humphreys' primary research interest has been in sodium metabolism and the pathophysiology of edema formation and salt-sensitive hypertension. He and his colleagues identified that rodent models of sodium retention like nephrotic syndrome, liver cirrhosis, and pregnancy are characterized by resistance to the natriuretic actions of atrial natriuretic peptide (ANP), and this in turn is caused by a heightened activity of Type V phosphodiesterase (PDE), which catabolizes cGMP formed normally in renal collecting duct cells when ANP interacts with its renal receptors. Inhibition of Type V PDE restores ANP responsiveness in these models. His group has also identified a novel hormonal system involved in normal sodium metabolism in rodents. It involves a peptide hormone gamma-melanocyte stimulating hormone (g-MSH) released from the pituitary ACTH precursor proopiomelanocortin. When animals are fed a high salt diet, g-MSH synthesis and secretion are up-regulated; it acts on the kidneys to increase sodium excretion, and on the brain to dampen down sympathetic excitation which occurs with high sodium intakes. When rodents have impaired ability to increase g-MSH secretion during ingestion of the high sodium diet, or lack the melanocortinr receptor with which it interacts, marked hypertension develops, and is accompanied by insulin resistance.
Dr. Humphreys has also done clinical research in these areas and has studied the occurrence of HIV-associated nephropathy in patients at San Francisco General Hospital. He participated in early studies measuring nitrogen balance in ESRD patients treated with hemodialysis, and was for a short time a site director for the Frequent Hemodialysis Network clinical trial.

Education
Residency, - School of Medicine, University of California, San Francisco
Honors and Awards
  • Leonard Share Award, Water and Electrolyte Homeostasis Section, American Physiological Society, 2019
  • John Alexander, MD Research Award, American Heart Association, 1999
  • Elected to American Clinical and Climatological Association, 1991
  • Alpha Omega Alpha Society, Case Western Reserve University, 1965
Publications
  1. Humphreys MH. Renal nerves and CKD: is renal denervation the answer? Volume 23 of Issue 7. Journal of the American Society of Nephrology : JASN 2012. PMID: 22677558


  2. Humphreys MH. The brain splits obesity and hypertension. Volume 17 of Issue 7. Nature medicine 2011. PMID: 21738154


  3. Humphreys MH, Ni XP, Pearce D. Cardiovascular effects of melanocortins. Volume 660 of Issue 1. European journal of pharmacology 2011. PMID: 21199648


  4. Sasser JM, Ni XP, Humphreys MH, Baylis C. Increased renal phosphodiesterase-5 activity mediates the blunted natriuretic response to a nitric oxide donor in the pregnant rat. Volume 299 of Issue 4. American journal of physiology. Renal physiology 2010. PMID: 20668100


  5. Chen S, Grigsby CL, Law CS, Ni X, Nekrep N, Olsen K, Humphreys MH, Gardner DG. Tonicity-dependent induction of Sgk1 expression has a potential role in dehydration-induced natriuresis in rodents. Volume 119 of Issue 6. The Journal of clinical investigation 2009. PMID: 19436108


  6. Ni XP, van Dijk C, Pearce D, Humphreys MH. Evidence for a noradrenergic mechanism causing hypertension and abnormal glucose metabolism in rats with relative deficiency of gamma-melanocyte-stimulating hormone. Volume 94 of Issue 8. Experimental physiology 2009. PMID: 19429645


  7. Ni XP, Humphreys MH. Abnormal glucose metabolism in hypertensive mice with genetically interrupted gamma-melanocyte stimulating hormone signaling fed a high-sodium diet. Volume 21 of Issue 12. American journal of hypertension 2008. PMID: 18802429


  8. Ni XP, Humphreys MH. Prevention of salt-induced hypertension by an analog of gamma-melanocyte-stimulating hormone in the rat. Volume 20 of Issue 8. American journal of hypertension 2007. PMID: 17679034


  9. Humphreys MH. Cardiovascular and renal actions of melanocyte-stimulating hormone peptides. Volume 16 of Issue 1. Current opinion in nephrology and hypertension 2007. PMID: 17143069


  10. Ni XP, Butler AA, Cone RD, Humphreys MH. Central receptors mediating the cardiovascular actions of melanocyte stimulating hormones. Volume 24 of Issue 11. Journal of hypertension 2006. PMID: 17053546


  11. Knight S, Snellen H, Humphreys M, Baylis C. Increased renal phosphodiesterase-5 activity mediates the blunted natriuretic response to ANP in the pregnant rat. Volume 292 of Issue 2. American journal of physiology. Renal physiology 2006. PMID: 17003222


  12. Ni XP, Bhargava A, Pearce D, Humphreys MH. Modulation by dietary sodium intake of melanocortin 3 receptor mRNA and protein abundance in the rat kidney. Volume 290 of Issue 3. American journal of physiology. Regulatory, integrative and comparative physiology 2005. PMID: 16195498


  13. Chen S, Ni XP, Humphreys MH, Gardner DG. 1,25 dihydroxyvitamin d amplifies type a natriuretic peptide receptor expression and activity in target cells. Volume 16 of Issue 2. Journal of the American Society of Nephrology : JASN 2004. PMID: 15590756


  14. Kalantar-Zadeh K, Block G, McAllister CJ, Humphreys MH, Kopple JD. Appetite and inflammation, nutrition, anemia, and clinical outcome in hemodialysis patients. Volume 80 of Issue 2. The American journal of clinical nutrition 2004. PMID: 15277149


  15. Ni XP, Safai M, Rishi R, Baylis C, Humphreys MH. Increased activity of cGMP-specific phosphodiesterase (PDE5) contributes to resistance to atrial natriuretic peptide natriuresis in the pregnant rat. Volume 15 of Issue 5. Journal of the American Society of Nephrology : JASN 2004. PMID: 15100365


  16. Kalantar-Zadeh K, Kopple JD, Humphreys MH, Block G. Comparing outcome predictability of markers of malnutrition-inflammation complex syndrome in haemodialysis patients. Volume 19 of Issue 6. Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 2004. PMID: 15069177


  17. Humphreys MH. Gamma-MSH, sodium metabolism, and salt-sensitive hypertension. Volume 286 of Issue 3. American journal of physiology. Regulatory, integrative and comparative physiology 2004. PMID: 14761863


  18. Kalantar-Zadeh K, Block G, Humphreys MH, McAllister CJ, Kopple JD. A low, rather than a high, total plasma homocysteine is an indicator of poor outcome in hemodialysis patients. Volume 15 of Issue 2. Journal of the American Society of Nephrology : JASN 2004. PMID: 14747392


  19. Kalantar-Zadeh K, Rodriguez RA, Humphreys MH. Association between serum ferritin and measures of inflammation, nutrition and iron in haemodialysis patients. Volume 19 of Issue 1. Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 2004. PMID: 14671049


  20. Mayan H, Ni XP, Almog S, Humphreys MH. Suppression of gamma-melanocyte-stimulating hormone secretion is accompanied by salt-sensitive hypertension in the rat. Volume 42 of Issue 5. Hypertension (Dallas, Tex. : 1979) 2003. PMID: 14568996


  21. Ni XP, Pearce D, Butler AA, Cone RD, Humphreys MH. Genetic disruption of gamma-melanocyte-stimulating hormone signaling leads to salt-sensitive hypertension in the mouse. Volume 111 of Issue 8. The Journal of clinical investigation 2003. PMID: 12697744


  22. Kalantar-Zadeh K, Block G, Humphreys MH, Kopple JD. Reverse epidemiology of cardiovascular risk factors in maintenance dialysis patients. Volume 63 of Issue 3. Kidney international 2003. PMID: 12631061


  23. Chen S, Cao L, Intengan HD, Humphreys M, Gardner DG. Osmoregulation of endothelial nitric-oxide synthase gene expression in inner medullary collecting duct cells. Role in activation of the type A natriuretic peptide receptor. Volume 277 of Issue 36. The Journal of biological chemistry 2002. PMID: 12082097


  24. Kalantar-Zadeh K, Kopple JD, Block G, Humphreys MH. Association among SF36 quality of life measures and nutrition, hospitalization, and mortality in hemodialysis. 2001. PMID: 11729250